Публикации

2022
IN SILICO IDENTIFICATION OF MULTI-TARGET LIGANDS AS PROMISING HIT COMPOUNDS FOR NEURODEGENERATIVE DISEASES DRUG DEVELOPMENT

P. Alov, H. Stoimenov, I. Lessigiarska, T. Pencheva, NikolayT. Tzvetkov, I. Pajeva, I. Tsakovska, International Journal of Molecular Sciences, 2022, 23, 13650.

2022
DIGITAL PILLS WITH INGESTIBLE SENSORS: PATENT LANDSCAPE ANALYSIS

O. Litvinova, E. Klager, Nikolay T. Tzvetkov, O. Kimberger, M. Kletecka-Pulker, H. Willschke, Atanas G. Atanasov, Pharmaceuticals 2022, 15, 1025.

2021
ADVANCES AND CHALLENGES IN CANCER TREATMENT AND NUTRACEUTICAL PREVENTION: THE POSSIBLE ROLE OF DIETARY PHENOLS IN BRCA REGULATION

Haroon Khan, Fabiana Labanca, Hammad Ullah, Yaseen Hussain, Nikolay T. Tzvetkov, Esra Küpeli Akkol, Luigi Milella, Phytochemistry Reviews 2021, 21, 385–400.

2025
REPURPOSING MAJOR METABOLITES OF LAMIACEAE FAMILY AS POTENTIAL INHIBITORS OF Α-SYNUCLEIN AGGREGATION TO ALLEVIATE NEURODEGENERATIVE DISEASES: AN IN SILICO APPROACH

Soham Bhattacharya, Neha Gupta, Adrish Dutta, Pijush Kanti Khanra, Ritesh Dutta, Jana Žiarovská, Dr Nikolay T Tzvetkov, Lucie Severová, Lenka Kopecká, Luigi Milella, Eloy Fernandez-Cusimamani, Frontiers in Pharmacology 2025, 16, 1519145.

2025
ENHANCING HUMAN GUT HEALTH: GLOBAL INNOVATIONS IN DYSBIOSIS MANAGEMENT

Reda El Boukhari, Maima Matin, Latifa Bouissane, Michał Ławiński, Oleh Lushchak, Rajeev K Singla, Michel‐Edwar Mickael, Jordi Mayneris‐Perxachs, Maria Eleni Grafakou, Shuhua Xu, Bowen Liu, Jiayi Guan, Andrzej Półtorak, Arkadiusz Szpicer, Agnieszka Wierzbicka, Nikolay T. Tzvetkov, Maciej Banach, Jarosław Olav Horbańczuk, Artur Jóźwik, Marco Cascella, Bairong Shen, Vasil Radoslavov Pirgozliev, Dongdong Wang, Olena Litvinova, Olga Adamska, Agnieszka Kamińska, Marcin Łapiński, Artur Stolarczyk, Ioana Berindan‐Neagoe, Luigi Milella, Andy Wai Kan Yeung, Prashanth Suravajhala, Anupam Bishayee, Ronan Lordan, Laszlo Barna Iantovics, Ricardo Lagoa, Monika Michalczuk, Jivko Stoyanov, A Douglas Kinghorn, Banaz Jalil, Wolfram Weckwerth, Bey Hing Goh, Meng‐Yao Li, Gyaneshwer Chaubey, Gian Luigi Russo, Sara Frazzini, Luciana Rossi, Maurizio Battino, Wei Jia, Qi Su, Xiaoqiang Ma, Judith M Rollinger, Simon K‐MR Rittmann, Helen Sheridan, John J. Walsh, Gerard Lizard, Tomasz M. Karpinski, Ana Sanches Silva, Jakub Piwowarski, Liwei Xie, Tai-Ping Fan, Franceska Giampieri, Adil El Midaoui, Ka-Hing Wong, Ren-You Gan, Ahmed Fatimi, Atanas G. Atanasov, iMeta 2025, e70028.

2024
Efficiency and safety of cannabinoid medical use: an analysis of discussions and observed trends on Instagram

Olena Litvinova, Bikash Baral, Thomas Wochele-Thoma, Maima Matin, Nikolay T. Tzvetkov, Olga Adamska, Agnieszka Kamińska, Marcin Łapiński, Artur Stolarczyk, Atanas G. Atanasov, Frontiers in Public Health 2024, 12, 1494018.

2024
IN SILICO EXPLORATION OF 4(Α-L-RHAMNOSYLOXY)-BENZYL ISOTHIOCYANATE: A PROMISING PHYTOCHEMICAL-BASED DRUG DISCOVERY APPROACH FOR COMBATING MULTI-DRUG RESISTANT STAPHYLOCOCCUS AUREUS

Soham Bhattacharya, Adrish Dutta, Pijush Kanti Khanra, Neha Gupta, Ritesh Dutta, Nikolay T. Tzvetkov, Luigi Milella, Maria Ponticelli, Computers in Biology and Medicine, 179, 108907.

2024
CRYSTAL STRUCTURES, MOLECULAR DOCKING AND IN VITRO INVESTIGATIONS OF TWO 4-SUBSTITUTED 2-(5,5-DIMETHYL-3-STYRYLCYCLOHEX-2-ENYLIDENE)MALONONITRILE DERIVATIVES AS POTENTIAL TOPOISOMERASE II INHIBITORS

Martina I. Peeva, Maya G. Georgieva, Aneliya A. Balacheva, Maria Ponticelli, Ivan P. Bogdanov, Tsonko Kolev, Luigi Milella, Hans-Georg Stammler, Nikolay T. Tzvetkov, Crystals, 14 (6), 496.

2024
WITHANIA SOMNIFERA (L.) DUNAL, A POTENTIAL SOURCE OF PHYTOCHEMICALS FOR TREATING NEURODEGENERATIVE DISEASES: A SYSTEMATIC REVIEW

Valentina Lerose, Maria Ponticelli, Nadia benedetto, Vittorio Carlucci, Ludovica Lela, Nikolay T. Tzvetkov, Luigi Milella, Plants 2024, 13(6), 771.

2024
NATURAL PRODUCT DRUG DISCOVERY AND DRUG DESIGN: TWO APPROACHES SHAPING NEW PHARMACEUTICAL DEVELOPMENT

Nikolay T. Tzvetkov, Kiril Kirilov, Maima Matin, Atanas G. Atanasov, Nephrology Dialysis Transplantation 2024, 39, 375–378.

2024
IN VITRO INVESTIGATION OF THE CYTOTOXIC AND ANTIPROLIFERATIVE EFFECTS OF HABERLEA RHODOPENSIS TOTAL EXTRACT: A COMPARATIVE STUDY

Martina I. Peeva, G. Georgieva, Maya, Aneliya A. Balacheva, Atanas Pavlov, Nikolay T. Tzvetkov, Cosmetics, 11 (2), 46.

2024
FAVIPIRAVIR VS. DEFERIPRONE: TAUTOMERIC, PHOTOPHYSICAL, IN VITRO BIOLOGICAL STUDIES, AND BINDING INTERACTIONS WITH SARS-COV-2-MPRO/ACE2

Nikolay T. Tzvetkov, Martina I. Peeva, Maya G. Georgieva, Vera Deneva, Aneliya A. Balacheva, Ivan P. Bogdanov, Maria Ponticelli, Luigi Milella, Kiril Kirilov, Maima Matin, Hans-Georg Stammler, Atanas G. Atanasov, Liudmil Antonov, Current Research in Biotechnology 2024, 7, 100176.

2023
AN INSIGHT INTO CITRUS MEDICA LINN.: A SYSTEMATIC REVIEW ON PHYTOCHEMICAL PROFILE AND BIOLOGICAL ACTIVITIES

Nadia Benedetto, Vittorio Carlucci, Immacolata Faraone, Ludovica Lela, Maria Ponticelli, Daniela Russo, Claudia Mangieri, Nikolay T. Tzvetkov, Luigi Milella, Plants 2023, 12(12), 2267.

2023
NEUROTENSIN (8–13) ANALOGS AS DUAL NTS1 AND NTS2 RECEPTOR LIGANDS WITH ENHANCED EFFECTS ON A MOUSE MODEL OF PARKINSON'S DISEASE

Toni Kühl, Maya G. Georgieva, Harald Hübner, Maria Lazarova, Matthias Vogel, Bodo Haas, Martina I. Peeva, Aneliya A. Balacheva, Ivan P. Bogdanov, Luigi Milella, Maria Ponticelli, Tsvetomir Garev, Immacolata Faraone, Roumyana Detcheva, Borislav Minchev, Polina Petkova-Kirova, Lyubka Tancheva, Reni Kalfin, Atanas G. Atanasov, Liudmil Antonov, Tamara I Pajpanova, Kiril Kirilov, Marcus Gastreich, Peter Gmeiner, Diana Imhof, Nikolay T. Tzvetkov, European Journal of Medicinal Chemistry 2023, 254, 115386.

2023
CYANIDIN-3-O-GLUCOSIDE AS A NUTRIGENOMIC FACTOR IN TYPE 2 DIABETES AND ITS PROMINENT IMPACT ON HEALTH

Iga Bartel, Magdalena Koszarska, Nina Strzałkowska, Nikolay T. Tzvetkov, Dongdong, Wang, Jarosław O Horbańczuk, Agnieszka Wierzbicka, Atanas G. Atanasov, Artur Jóźwik, International Journal of Molecular Sciences 2023, 24(11), 9765.

2023
BIBLIOMETRIC ANALYSIS AND EVIDENCE OF CLINICAL EFFICACY AND SAFETY OF DIGITAL PILLS

Olena Litvinova, Elisabeth Klager, Andy Wai Kan Yeung, Nikolay T. Tzvetkov, Oliver Kimberger, Maria Kletecka-Pulker, Harald Willschke, Atanas G. Atanasov, Frontiers in Pharmacology 2023, 14, 1023250.

2022
SR-BI AS A TARGET OF NATURAL PRODUCTS AND ITS SIGNIFICANCE IN CANCER

D. Wang, J. Huang, T. Gui, Y. Yang, T. Feng, N.T. Tzvetkov, T. Xu, Z. Gai, Y. Zhou, J. Zhang, A.G. Atanasov, Seminars in Cancer Biology 2022, 80, 18–38.

2012
REGIOSELECTIVE SYNTHESIS OF 7, 8-DIHYDROIMIDAZO [5, 1-C][1, 2, 4] TRIAZINE-3, 6 (2H, 4H)-DIONE DERIVATIVES: A NEW DRUG-LIKE HETEROCYCLIC SCAFFOLD

Nikolay T. Tzvetkov, Harald Euler, Christa E. Müller, Beilstein Journal of Organic Chemistry 2012, 8(1), 1584–1593.

2012
FACILE SYNTHESIS OF 5-AMINO-AND 7-AMINO-6-AZAOXINDOLE DERIVATIVES

Nikolay T. Tzvetkov, Christa E. Müller, Tetrahedron Letters 2012, 53(42), 5597–5601.

2021
NATURAL PRODUCTS IN DRUG DISCOVERY: ADVANCES AND OPPORTUNITIES

A.G. Atanasov, S.B. Zotchev, V.M. Dirsch, The International Natural Product Sciences Taskforce, N.T. Tzvetkov, C.T. Sapuran, Nature Reviews Drug Discovery 2021, 20, 200–216.

2021
VASCUPROTECTIVE EFFECTS OF GINGER (ZINGIBER OFFICINALE ROSCOE) AND UNDERLYING MOLECULAR MECHANISMS

C. Li, J. Li, F. Jiang, N.T. Tzvetkov, J.O. Horbañczuk, Y. Li, A.G. Atanasov D. Wang, Food & Function 2021, 12(5), 1897–1913.

2021
REACTIVE OXYGEN SPECIES AND THEIR IMPACT IN NEURODEGENERATIVE DISEASES: LITERATURE LANDSCAPE ANALYSIS

A.W.K. Yeung, N.T. Tzvetkov, M.G. Georgieva, I.V. Ognyanov, K. Kordos, A. Jozwik, T. Kühl, G. Perry, M.C. Petralia, E. Mazzon, A.G. Atanasov, Antioxidants & Redox Signaling 2021, 34(5), 402–420.

2020
PREVENTIVE EFFECT OF A POLYPHENOL-RICH EXTRACT FROM GERANIUM SANGUINEUM L. ON HEPATIC DRUG METABOLISM IN INFLUENZA INFECTED MICE

Silviya Abarova, Lyubka Tancheva, Rumen Nikolov, Julia Serkedjieva, Elitsa Pavlova, Alessia Bramanti, Ferdinando Nicoletti, Nikolay T. Tzvetkov, Scientia Pharmaceutica 2020, 88(4), 45.

2020
THE ETHNOPHARMACOLOGICAL LITERATURE: AN ANALYSIS OF THE SCIENTIFIC LANDSCAPE

Andy Wai Kan Yeung, Michael Heinrich, Anake Kijjoa, Nikolay T. Tzvetkov, Atanas G. Atanasov, Journal of Ethnopharmacology 2020, 250, 112414.

2020
ETHNOPHARMACOLOGICAL APPLICATIONS TARGETING ALCOHOL ABUSE: OVERVIEW AND OUTLOOK

Laxman Singh, Tanuj Joshi, Devesh Tewari, Javier Echeverría, Andrei Mocan, Archana N Sah, Nikolay T. Tzvetkov, Zheng Feei Ma, Yeong Yeh Lee, Piotr Poznański, Mariusz Sacharczuk, Artur Jóźwik, Jarosław O Horbańczuk, Joanna Feder-Kubis, Atanas G. Atanasov, Frontiers in Pharmacology 2020, 10, 481687.

2020
THE SIGNIFICANCE OF NATURAL PRODUCT DERIVATIVES AND TRADITIONAL MEDICINE FOR COVID-19

D. Wang, J. Huang, A.W.K. Yeung, N.T. Tzvetkov, J.O. Horbañczuk, H. Willschke, Z. Gai, A.G. Atanasov, Processes 2020, 8, 937.

2020
LIGNANS: QUANTITATIVE ANALYSIS OF THE RESEARCH LITERATURE

A.W.K. Yeung, N.T. Tzvetkov, A.A. Balacheva, M.G. Georgieva, R.-Y. Gan, A. Jozwik, B. Pyzel, J.O. Horbañczuk, E. Novellino, A. Durazzo, M. Lucarini, E. Camilli, E.B. Souto, A.G. Atanasov, A. Santini, Frontiers in Pharmacology 2020, 11, Article 37.

2020
NEUROPROTECTIVE MECHANISMS OF THREE NATURAL ANTIOXIDANTS ON A RAT MODEL PARKINSON´S DISEASE: A COMPARATIVE STUDY

L.P. Tancheva, M.I. Lazarova, A.V. Alexandrova, S.T. Dragomanova, F. Nicoletti, E.R. Tzvetanova, Y.K. Hodzhev, R.E. Kalfin, S.A. Miteva, A. Santini, E. Mazzon, N.T. Tzvetkov, A.G. Atanasov, Antioxidants 2020, 9(1), 49.

2020
NEUROTENSINS AND THEIR THERAPEUTIC POTENTIAL: RESEARCH FIELD STUDY

A.W.K. Yeung, M.G. Georgieva, K. Kirilov, A.A. Balacheva, M.I. Peeva, O.K. Horbañczuk, J.O. Horbañczuk, M. Lucarini, A. Durazzo, A. Santini, E.B. Souto, T.I. Pajpanova, L. Milella, A.G. Atanasov, N.T. Tzvetkov, Future Medicinal Chemistry 2020, 12(19), 1779–1803.

2019
CURRENT RESEARCH IN BIOTECHNOLOGY: EXPLORING THE BIOTECH FOREFRONT

Andy Wai Kan Yeung, Nikolay T. Tzvetkov, Vijai K Gupta, Subash C Gupta, Gorka Orive, Günther K Bonn, Bernd Fiebich, Anupam Bishayee, Thomas Efferth, Jianbo Xiao, Ana Sanches Silva, Gian Luigi Russo, Maria Daglia, Maurizio Battino, Ilkay Erdogan Orhan, Ferdinando Nicoletti, Michael Heinrich, Bharat Bhushan Aggarwal, Marc Diederich, Maciej Banach, Wolfram Weckwerth, Rudolf Bauer, George Perry, Edward A Bayer, Lukas A Huber, Jean-Luc Wolfender, Robert Verpoorte, Francisco A Macias, Michael Wink, Marc Stadler, Simon Gibbons, Alejandro Cifuentes, Elena Ibanez, Gérard Lizard, Rolf Müller, Michael Ristow, Atanas G. Atanasov, Current Research in Biotechnology 2019, 1, 34–40.

2019
MOLECULAR NEUROSCIENCE AT ITS “HIGH”: BIBLIOMETRIC ANALYSIS OF THE MOST CITED PAPERS ON ENDOCANNABINOID SYSTEM, CANNABIS AND CANNABINOIDS

Andy Wai Kan Yeung, Nikolay T. Tzvetkov, Nicolas Arkells, Luigi Milella, Adrian M Stankiewicz, Łukasz Huminiecki, Olaf K Horbanczuk, Atanas G. Atanasov, Journal of Cannabis Research 2019, 1, 1–13.

2019
TARGETING FOAM CELL FORMATION IN ATHEROSCLEROSIS: THERAPEUTIC POTENTIAL OF NATURAL PRODUCTS

D. Wang, Y. Yang, Y. Lei, N.T. Tzvetkov, Y. Liu, A.W.K Yeung, S. Xu, A.G. Atanasov, Pharmacological Reviews 2019, 71(4), 596– 670.

2019
CARBOXAMIDES VS. METHANIMINES: CRYSTAL STRUCTURES, BINDING INTERACTIONS, PHOTOPHYSICAL STUDIES, AND BIOLOGICAL EVALUATION OF (INDAZOLE-5-YL)METHANIMINES AS MONOAMINE OXIDASE B AND ACETYLCHOLONESTERASE INHIBITORS

N.T. Tzvetkov, H.-G. Stammler, M.G. Georgieva, D. Russo, I. Faraone, A.A. Balacheva, S. Hristova, A.G. Atanasov, L. Milella, L. Antonov, M. Gastreich, European Journal of Medicinal Chemistry 2019, 179, 404–422.

2019
(PYRROLO-PYRIDIN-5- YL)BENZAMIDES: BBB PERMEABLE MONOAMINE OXIDASE B INHIBITORS WITH NEUROPROTECTIVE EFFECT ON CORTICAL NEURONS

N.T. Tzvetkov, H.-G. Stammler , S. Hristova, A.G. Atanasov, L. Antonov, European Journal of Medicinal Chemistry 2019, 162, 793–809.

2019
MONOAMINE OXIDASES (MAOS) AS PRIVILEGED MOLECULAR TARGETS IN NEUROSCIENCE: RESEARCH LITERATURE ANALYSIS

A.W.K. Yeung, M. Georgieva, A.G. Atanasov, N.T. Tzvetkov, Frontiers in Molecular Neuroscience 2019, 12, Article 413.

2019
ANTIOXIDANTS: SCIENTIFIC LITERATURE LANDSCAPE

A.W.K. Yeung, N.T. Tzvetkov, O.S. El-Tawil, S.G. Bungau, M.M. Abdel-Daim, A.G. Atanasov, Oxidative Medicine and Cellular Longevity 2019, Article ID 8278454.

2018
VASCULOPROTECTIVE EFFECTS OF POMEGRANATE (PUNICA GRANATUM L.)

Dongdong Wang, Cigdem Özen, Ibrahim M Abu-Reidah, Sridevi Chigurupati, Jayanta Kumar Patra, Jarosław O. Horbanczuk, Artur Jóźwik, Nikolay T. Tzvetkov, Pavel Uhrin, Atanas G. Atanasov, Frontiers in Pharmacology 2018, 9, 544.

2018
NATURAL PRODUCT-BASED MULTITARGET LIGANDS FOR ALZHEIMER’S DISEASE TREATMENT?

N.T. Tzvetkov, A.G. Atanasov, Future Medicinal Chemistry 2018, 10, 1745–1748.

2018
WHEN NEUROSCIENCE MEETS PHARMACOLOGY: A NEUROPHARMACOLOGY LITERATURE ANALYSIS

A.W.K. Yeung, N.T. Tzvetkov, A.G. Atanasov, Frontiers in Neuroscience 2018, 12, Article 852.

2018
PHYTOCHEMICALS AS POTENT MODULATOES AF AUTOPHAGY FOR CANCER THERAPY

M.A. Moosavi, A. Hghi, M. Rahmati, H. Taniguchi, A. Mocan, J. Echeverria, V.K.Gupta, N.T. Tzvetkov, A.G. Atanasov, Cancer Letters 2018, 424, 46–69.

2018
AUTOPHAGY AND ALZHEIMER’S DISEASE: FROM MOLECULAR MECHANISMS TO THERAPEUTIC IMPLICATIONS

Md. Uddin, A. Stachowiak, A.A. Mamun, N.T. Tzvetkov, S. Takeda, A.G. Atanasov, L.B. Bergantin, M.M. Abdel-Daim, A.M. Stankiewicz, Frontiers in Aging Neuroscience 2018, 10, Article 4.

2018
ETHNOPHARMACOLOGICAL APPROACHES FOR DEMENTIA THERAPY AND SIGNIFICANCE OF NATURAL PRODUCTS AND HERBAL DRUGS

D. Tewari, A.M. Stankiewicz, A. Mocan, A.N. Sah, N.T. Tzvetkov, L. Huminiecki, J.O. Horbañczuk, A.G. Atanasov, Frontiers in Aging Neuroscience 2018, 10, Article 3.

2018
PREVENTIVE EFEFCT OF TWO NEW NEUROTENSIN ANALOGUES ON PARKINSON’S DISEASE RAT MODEL

M. Lazarova, A. Popatanasov, R. Klissurov, S. Stoeva, T. Pajpanova, R. Kalfin, L. Tancheva, Journal of Molecular Neuroscience 2018, 66, 552–560.

2018
VASCULAR SMOOTH MUSCLE CELL PROLIFERATION AS A THERAPEUTIC TARGET. PART 2: NATURAL PRODUCTS INHIBITING PROLIFERATION

P. Uhrin, D. Wang, A. Mocan, B. Waltenberger, J.M. Breuss, D. Tewari, J. Mihaly-Bison, L. Huminiecki, R.R. Starzyñski, N.T. Tzvetkov, J. Horbañczuk, A.G. Atanasov, Biotechnology Advances 2018, 36, 1608–1621.

2018
VASCULAR SMOOTH MUSCLE CELL PROLIFERATION AS A THERAPEUTIC TARGET. PART 1: MOLECULAR TARGETS AND PATHWAYS

P. Uhrin, D. Wang, A. Mocan, B. Waltenberger, J.M. Breuss, D. Tewari, J. Mihaly-Bison, L. Huminiecki, R.R. Starzyñski, N.T. Tzvetkov, J. Horbañczuk, A.G. Atanasov, Biotechnology Advances 2018, 36, 1586–1607.

2017
TAUTOMERISM OF N-(3, 4-DICHLOROPHENYL)-1H-INDAZOLE-5-CARBOXAMIDE–A NEW SELECTIVE, HIGHLY POTENT AND REVERSIBLE MAO-B INHIBITOR

Nikolay T. Tzvetkov, Hans-Georg Stammler, Liudmil Antonov, Journal of Molecular Structure 2017, 1149, 273–281.

2017
CRYSTAL STRUCTURES, BINDING INTERACTIONS, AND ADME EVALUATION OF BRAIN PENETRANT N-SUBSTITUTED CARBOXAMIDES AS SUBNANOMOLAR, SELECTIVE MONOAMINE OXIDASE B AND DUAL MAO-A/B INHIBITORS

N.T. Tzvetkov, H.-G. Stammler, B. Neumann, S. Hristova, L. Antonov, M. Gastreich, European Journal of Medicinal Chemistry 2017, 127, 470–492.

2016
A SIMPLE APPROACH TO MULTIFUNCTIONALIZED N1-ALKYLATED 7-AMINO-6-AZAOXINDOLE DERIVATIVES USING THEIR IN SITU STABILIZED TAUTOMER FORM

Nikolay T. Tzvetkov, Beate Neumann, Hans-Georg Stammler, Liudmil Antonov, Tetrahedron 2016, 72(41), 6455–6466.

2014
NTERACTION OF METHIONINE – ENKEPHALINS WITH RAFT-FORMING LIPIDS: MONOLAYERS AND BAM EXPERIMENTS

A. Tsanova, A. Jordanova, T Dzimbova, T. Pajpanova, E. Golovinsky, Z. Lalchev, Amino Acids 2014, 46, 1159–1168.

2014
KYOTORPHIN ANALOGUES CONTAINING UNNATURAL AMINO ACIDS: SYNTHESIS, ANALGESIC ACTIVITY AND COMPUTER MODELING OF THEIR INTERACTIONS WITH Μ-RECEPTOR

T. Dzimbova, A. Bocheva, T. Pajpanova, Medicinal Chemistry Research 2014, 23, 3694–3704.

2014
INDAZOLE- AND INDOLE-5-CARBOXAMIDES: SELECTIVE AND REVERSIBLE MONOAMINE OXIDASE B INHIBITORS WITH SUBNANOMOLAR POTENCY

N.T. Tzvetkov, S. Hinz, P. Küppers, M. Gastreich, C.E. Müller, Journal of Medicinal Chemistry 2014, 57, 6679–6703.

2024
AVPI analogs and conjugates: Molecular docking studies and in vitro biological evaluation

Maya G. Georgieva, Silvia G. Mihaylova, Aneliya A. Balacheva, Antoaneta Z. Tsvetkova, Tamara I. Pajpanova, Nikolay T. Tzvetkov, Current Research in Biotechnology 2024, 8, 100246.

2024
Effects of Ginger (Zingiber officinale) on the Hallmarks of Aging

Maima Matin, Tanuj Joshi, Dongdong Wang, Nikolay T. Tzvetkov, Farhan Bin Matin, Agnieszka Wierzbicka, Artur Jóźwik, Jarosław Olav Horbańczuk, Atanas G. Atanasov, Biomolecules 2024, 14(8), 940.

2024
Insight into the Interaction of Humulus lupulus L. Specialized Metabolites and Gastrointestinal Bitter Taste Receptors: In Vitro Study in STC-1 Cells and Molecular Docking

Ludovica Lela, Maria Ponticelli, Vittorio Carlucci, Jan F Stevens, Immacolata Faraone, Nikolay T. Tzvetkov, Luigi Milella, Journal of Natural Products 2024, 87(8), 2021–2033.

2022
ADVANCES AND CHALLENGES IN CANCER TREATMENT AND NUTRACEUTICAL PREVENTION: THE POSSIBLE ROLE OF DIETARY PHENOLS IN BRCA REGULATION

H. Khan, F. Labanca, H. Ullah, Y. Hussain, Nikolay T. Tzvetkov, E. K. Akkol, Luigi Milella, Phytochemistry Reviews 2022, 21, 385–400.